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Posaconazole takawaenga

  • (5R-cis)-Toluene-4-sulfonic acid 5-(2,4-difluorophenyl)-5-(1H-1,2,4-triazol-1-yl)methyltetrahydrofuran-3-ylmethyl ester

    (5R-cis)-Toluene-4-sulfonic acid 5-(2,4-difluorophenyl)-5-(1H-1,2,4-triazol-1-yl)methyltetrahydrofuran-3-ylmethyl ester

    Nga Ahuatanga matū me te tinana

    Posaconazole takawaenga.

    Ko Posaconazole, i whakarewahia i te UK, ko te mema hou o te akomanga azole o nga kaihoko antifungal kia tae ki te maakete.E tohuhia ana mo te maimoatanga me te aukati i te tini o nga mate harore invasive, tae atu ki te aspergillosis, fusariosis, chromoblastomycosis, mycetoma, me te coccidiomycosis i roto i nga turoro e whakakeke ana, e kore e manawanui ki te rongoa paerewa me te amphotericin B me/ranei itraconazole.I roto i te US, ka whakaaetia mo te aukati i nga mate urutomo Aspergillus me Candida ki nga turoro 13 tau te pakeke e tino tupono ana ki te whakawhanake i enei mate na te kaha o te mate mate.I tua atu, kua whakaaetia mo te maimoatanga o te candidiasis oropharyngeal.Ko te Posaconazole he nui ake te mahi a te Posaconazole ki runga ake i etahi atu mema o te azole antifungals.I tua atu i te kaha kaha ki te aukati i nga keehi o te aspergillosis me te Candida-atete ki te fluconazole, e whakaatu ana i te mahi ki a Zygomycetes.

    Mena kei te pirangi koe ki a maatau hua, he patai ranei, tena koa whakapiri mai ki a maatau!

    Ko nga hua kei raro i te patent ka tukuna mo te kaupapa R&D anake.

  • 2-[(1S,2S)-1-ethyl-2-bezyloxypropyl]-2,4-dihydro-4-[4-[4-(4-hydroxyphenyl)-1-piperazinyl]phenyl]- 3H-1,2 ,4-Triazol-3-one

    2-[(1S,2S)-1-ethyl-2-bezyloxypropyl]-2,4-dihydro-4-[4-[4-(4-hydroxyphenyl)-1-piperazinyl]phenyl]- 3H-1,2 ,4-Triazol-3-one

    Nga Ahuatanga matū me te tinana

    Takawaenga i roto i te faaineineraa o Posaconazole.

    Mena kei te pirangi koe ki a maatau hua, he patai ranei, tena koa whakapiri mai ki a maatau!

    Ko nga hua kei raro i te patent ka tukuna mo te kaupapa R&D anake.