page_banner

I te Paenga-whāwhā 15, 2022, i oti te hanga pairati o te whakakai matua Lecardipine hydrochloride i te wa kotahi, a ko te kaha whakaputa o naianei he 5Mt/marama.

I te Paenga-whāwhā 15, 2022, i oti te hanga pairati o te whakakai matua Lecardipine hydrochloride i te wa kotahi, a ko te kaha whakaputa o naianei he 5Mt/marama.
Ingoa Ingarihi:Lercanidipine hydrochloride
Ingoa matū:1,4-Dihydro-2,6-dimethyl-4-(3-nitrophenyl) -3,5-pyridinedicarboxylic acid 2- [(3,3-di phenylpropyl)methylamino]-l,l-dimethylethyl methyl ester hydrochloride.

Nama CAS: 132866-11-6
Taupānga:Mo te maimoatanga o te rongoa Lecardipine hydrochloride, kare he paanga kino ki te huka toto me nga taumata lipid, a he kaha te awenga antihypertensive.

Te maakete:
Neke atu i te 200 miriona nga turoro mate pukupuku i Haina, a he 10 miriona nga turoro mate pukupuku hou i ia tau, ko te nuinga o enei kaore i raro i te mana whakahaere, na te nui o te mate o nga mate whakaheke toto penei i te whiu, me te mate o te tau i Haina I roto i te 3 miriona nga turoro me te mate mate pukupuku, 50% e pa ana ki te whakaheke toto, a ko te utu o te tau mo te maimoatanga mate pukupuku e tata ana ki te 309.8 piriona yuan.Ko te take o te ngoikoretanga o te whakahaere ehara i te mea ko te mohiotanga o nga turoro ki te whakaheke toto me ona raruraru me whakapai ake, engari he maha nga turoro e hiahia ana ki te tango i nga rongoa mo te wa katoa, he ngoikore te hanganga ture, kaore e taea te tango rongoa i ia ra Heoi, e whakaatu ana hoki tenei Ko te maakete tarukino antihypertensive ka kaha te tipu.Ka whakatauritea ki nga raau taero rite, ko te locarbodipine hydrochloride he kaha te kowhiringa o te toto.Ko tana taonga lipophilic ahurei ka puhoi, ka mau tonu te paanga antihypertensive Ko te paanga atherogenic, he pai rawa mo nga turoro whakaheke toto me te atherosclerosis, he nui te uara tono haumanu me te maakete whanui.

Mahi rongoa:
Ko te Lecardipine he whakatipuranga hou o te dihydropyridine calcium channel group hysteresis agent, me te kaha o te whiriwhiringa vascular, te kaha ngawari, te kaha antihypertensive, te wa mahi roa, te iti o te kino inotropic me etahi atu.I kitea e nga rangahau in vitro ko te locarbodipine he whakangawari tika ki nga uaua maeneene vascular, na reira he kaha te hua antihypertensive i roto i te vivo, engari he iti te paanga o te ngakau me te whakaputa ngakau.Na te nui o te ira hydrophobic me te kaha o te wairewa lipid, ka tere te tohatoha o te locarbodipine ki nga kopa me nga whekau i muri i te urunga ki roto i te tinana, ka piri tata ki te kirikiri o nga uaua ngongo ngongo, me te tuku ata.Na reira, ahakoa he wa poto te whakakorenga o te serum o tenei tarukino mo te haurua o te kore, he roa te hua.


Te wa tuku: Apr-15-2022